Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors
August 29th, 2016 by Tinghu Zhang
Nature Chemical Biology 12, 876 (2016). doi:10.1038/nchembio.2166
Authors: Tinghu Zhang, Nicholas Kwiatkowski, Calla M Olson, Sarah E Dixon-Clarke, Brian J Abraham, Ann K Greifenberg, Scott B Ficarro, Jonathan M Elkins, Yanke Liang, Nancy M Hannett, Theresa Manz, Mingfeng Hao, Bartlomiej Bartkowiak, Arno L Greenleaf, Jarrod A Marto, Matthias Geyer, Alex N Bullock, Richard A Young & Nathanael S Gray