Long Residence Time Inhibition of EZH2 in Activated Polycomb Repressive Complex 2

December 31st, 2013 by Glenn S. Van Aller, Melissa Baker Pappalardi, Heidi M. Ott, Elsie Diaz, Martin Brandt, Benjamin J. Schwartz, William H. Miller, Dashyant Dhanak, Michael T. McCabe, Sharad K. Verma, Caretha L. Creasy, Peter J. Tummino and Ryan G. Kruger

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ACS Chemical Biology
DOI: 10.1021/cb4008748